Molecule Details
InChIKeyUPJFBUSSMBUXBJ-UHFFFAOYSA-N
Compound Name3-amino-N-(2,6-difluorobenzyl)-6-(1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-5-(oxazol-2-yl)pyrazine-2-carboxamide
Canonical SMILESCn1cc(-c2nc(C(=O)NCc3c(F)cccc3F)c(N)nc2-c2ncco2)ccc1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.46
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29275 ADORA2B Homo sapiens Human PF00001 8.8 IC50 ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 8.7 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.8 IC50 ChEMBL;BindingDB