Molecule Details
InChIKeyUOYOWVPLBRMQFZ-UHFFFAOYSA-N
Compound NameN-(4-((4-methylpiperazin-1-yl)methyl)phenyl)-4-((6-methylthieno[2,3-d]pyrimidin-4-yl)amino)-1H-pyrazole-3-carboxamide
Canonical SMILESCc1cc2c(Nc3c[nH]nc3C(=O)Nc3ccc(CN4CCN(C)CC4)cc3)ncnc2s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.98
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 9.4 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 8.8 IC50 ChEMBL;BindingDB
P78396 CCNA1 Homo sapiens Human PF02984 PF00134 PF16500 8.8 IC50 ChEMBL