Molecule Details
InChIKeyUOMPPOVQMYNXST-KDOFPFPSSA-N
Compound NameN-[4-[(2R,3S)-3-amino-2-methylpiperidin-1-yl]-3-pyridinyl]-2-(2,6-difluorophenyl)imidazo[1,5-b]pyridazin-7-amine
Canonical SMILESC[C@@H]1[C@@H](N)CCCN1c1ccncc1Nc1ncc2ccc(-c3c(F)cccc3F)nn12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.73
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 10.0 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 9.5 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 6.7 IC50 ChEMBL