Molecule Details
InChIKeyUNUTTXCETMYXRD-UHFFFAOYSA-N
Compound NameN-(4-Methyl-3-(3-methyl-1H-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(2-oxo-3,4-dihydroquinolin-1(2H)-yl)acetamide
Canonical SMILESCc1n[nH]c(-c2c(C)csc2NC(=O)CN2C(=O)CCc3ccccc32)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.6
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB