Molecule Details
InChIKeyUNTVUXKLSQXPLR-NWTJGDGASA-N
Compound Name(13S,17S)-17-[di(propan-2-yl)carbamoyl]-13-methyl-8,9,11,12,14,15,16,17-octahydrocyclopenta[a]phenanthrene-3-carboxylic acid
Canonical SMILESCC(C)N(C(=O)[C@H]1CCC2C3C=Cc4cc(C(=O)O)ccc4C3CC[C@@]21C)C(C)C
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.52
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.5 pIC50 TTD_MultiTarget
P31639 SLC5A2 Homo sapiens Human PF00474 7.5 pIC50 TTD_MultiTarget