Molecule Details
InChIKeyUNSAZGGWYRHTHJ-UHFFFAOYSA-N
Compound Name6-[2-(dimethylamino)ethyl]-2-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]-7H-pyrrolo[3,4-b]pyridin-5-one
Canonical SMILESCc1nc2c(F)cc(-c3nc(Nc4ccc5c(n4)CN(CCN(C)C)C5=O)ncc3F)cc2n1C(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB