Molecule Details
InChIKeyUNQRXDNHUDKYHT-UHFFFAOYSA-N
Compound Name2-[2-[2-[2-[Carboxymethyl-[2-oxo-2-[2-(4-sulfamoylphenyl)hydrazinyl]ethyl]amino]ethoxy]ethoxy]ethyl-[2-oxo-2-[2-(4-sulfamoylphenyl)hydrazinyl]ethyl]amino]acetic acid
Canonical SMILESNS(=O)(=O)c1ccc(NNC(=O)CN(CCOCCOCCN(CC(=O)O)CC(=O)NNc2ccc(S(N)(=O)=O)cc2)CC(=O)O)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.68
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 6.7 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 6.7 pIC50 TTD_MultiTarget