Molecule Details
InChIKeyUNEVEWKTGHFQJP-UHFFFAOYSA-N
Compound Name7-[Amino-(4-chlorophenyl)-(3-methylimidazol-4-yl)methyl]-10-(3-chlorophenyl)-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5,7,9(13),10-tetraen-12-one
Canonical SMILESCn1cncc1C(N)(c1ccc(Cl)cc1)c1cc2c3c(c1)c(-c1cccc(Cl)c1)cc(=O)n3CCO2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.8
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.8 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.8 IC50 ChEMBL