Molecule Details
InChIKeyUNEUBPFDOWMHSM-UHFFFAOYSA-N
Compound Name2-[Bis[2-[carboxymethyl-[2-oxo-2-[2-(4-sulfamoylphenyl)hydrazinyl]ethyl]amino]ethyl]amino]acetic acid
Canonical SMILESNS(=O)(=O)c1ccc(NNC(=O)CN(CCN(CCN(CC(=O)O)CC(=O)NNc2ccc(S(N)(=O)=O)cc2)CC(=O)O)CC(=O)O)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.57
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 6.7 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 6.7 pIC50 TTD_MultiTarget
P22748 CA4 Homo sapiens Human PF00194 6.4 Ki ChEMBL;BindingDB