Molecule Details
InChIKeyUNCZUEUPSJKHGB-UHFFFAOYSA-N
Compound Name3-(2,4-Dimethylpyrido[2',3':3,4]pyrazolo[1,5-a]pyrimidin-3-yl)-N-(3-(methylthio)phenyl)propanamide
Canonical SMILESCSc1cccc(NC(=O)CCc2c(C)nc3c4cccnc4nn3c2C)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.02
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9BZ23 PANK2 Homo sapiens Human PF03630 7.0 IC50 ChEMBL;BindingDB
Q9H999 PANK3 Homo sapiens Human PF03630 7.0 IC50 ChEMBL;BindingDB
Q8TE04 PANK1 Homo sapiens Human PF03630 7.0 IC50 ChEMBL;BindingDB