Molecule Details
InChIKeyULQVOSFGFYDDOI-HXUWFJFHSA-N
Compound NameN-(2-aminophenyl)-4-[[(4S)-4-pyridin-3-yl-4,5-dihydro-1,3-oxazol-2-yl]sulfanylmethyl]benzamide
Canonical SMILESNc1ccccc1NC(=O)c1ccc(CSC2=N[C@@H](c3cccnc3)CO2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O15379 HDAC3 Homo sapiens Human PF00850 7.2 IC50 ChEMBL;BindingDB
Q9Y618 NCOR2 Homo sapiens Human PF15784 PF00249 7.2 IC50 ChEMBL
Q92769 HDAC2 Homo sapiens Human PF00850 6.2 IC50 ChEMBL;BindingDB