Molecule Details
InChIKeyUKUBGLJCBLBBTL-UHFFFAOYSA-N
Compound Name3-[4-(3-Amino-1,2-benzothiazol-4-yl)phenyl]-1-[3-(trifluoromethyl)phenyl]urea
Canonical SMILESNc1nsc2cccc(-c3ccc(NC(=O)Nc4cccc(C(F)(F)F)c4)cc3)c12
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.61
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P35968 KDR Homo sapiens Human PF07679 PF00047 PF13895 PF22971 PF07714 PF21339 PF17988 PF22854 6.6 IC50 ChEMBL;BindingDB
Q02161 RHD Homo sapiens Human PF00909 6.6 pIC50 TTD_MultiTarget