Molecule Details
InChIKeyUKNGIFKYRYBARW-UHFFFAOYSA-N
Compound Name4-(4-(Pyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-ylamino)benzamide
Canonical SMILESNC(=O)c1ccc(Nc2nccc(-c3cnn4ncccc34)n2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.77
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.8 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 7.8 pIC50 TTD_MultiTarget
P49841 GSK3B Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB