Molecule Details
InChIKeyUKGCAEYEQULSSN-UHFFFAOYSA-N
Compound NameN-[4-(1-acetylpiperidin-4-yl)-2-(cyclohexen-1-yl)phenyl]-5-cyano-1H-imidazole-2-carboxamide
Canonical SMILESCC(=O)N1CCC(c2ccc(NC(=O)c3ncc(C#N)[nH]3)c(C3=CCCCC3)c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P07333 CSF1R Homo sapiens Human PF00047 PF25305 PF07714 8.7 IC50 ChEMBL;BindingDB
P10721 KIT Homo sapiens Human PF00047 PF07714 7.2 IC50 ChEMBL;BindingDB