Molecule Details
InChIKeyUKFKDADMCDDXJG-HGBJFFEJSA-N
Canonical SMILESCCOc1cc([C@]2(c3nncn3C)C[C@@H](C)C2)cc(N2Cc3c(cc(CNC4(C)CCC4)cc3C(F)(F)F)C2=O)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.46
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P06239 LCK Homo sapiens Human PF07714 PF00017 PF00018 8.5 IC50 BindingDB
Q13191 CBLB Homo sapiens Human PF02262 PF02761 PF02762 PF00097 8.4 IC50 ChEMBL