Molecule Details
InChIKeyUKAGZEMTXTYYHX-MRXNPFEDSA-N
Compound Name(3R)-1-[3-[5-(1-methylpyrazol-4-yl)-1H-pyrazolo[3,4-c]pyridin-3-yl]phenyl]piperidin-3-amine
Canonical SMILESCn1cc(-c2cc3c(-c4cccc(N5CCC[C@@H](N)C5)c4)n[nH]c3cn2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.28
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.5 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.4 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.9 Ki ChEMBL;BindingDB