Molecule Details
InChIKeyUJQKNBFBUSXTSO-CMPLNLGQSA-N
Canonical SMILESCC(C)c1n[nH]c2c(=O)[nH]c(C[C@@H]3CCCC[C@H]3Nc3ncc(C(=O)O)c(C(F)(F)F)n3)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O76083 PDE9A Homo sapiens Human PF00233 8.2 IC50 ChEMBL
O76074 PDE5A Homo sapiens Human PF01590 PF00233 6.4 IC50 ChEMBL;BindingDB