Molecule Details
InChIKeyUJAZDXIAIGDQSX-UHFFFAOYSA-N
Compound Name6-Ethyl-3-[3-(4-methoxycarbonyl-4-phenyl-piperidin-1-yl)-propylcarbamoyl]-4-(4-nitro-phenyl)-2-oxo-1,2,3,4-tetrahydro-pyrimidine-5-carboxylic acid methyl ester
Canonical SMILESCCC1=C(C(=O)OC)C(c2ccc([N+](=O)[O-])cc2)N(C(=O)NCCCN2CCC(C(=O)OC)(c3ccccc3)CC2)C(=O)N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.86
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB