Molecule Details
InChIKeyUIRLFLOVKAOFEX-UHFFFAOYSA-N
Compound NameBenzeneacetamide, N-(4-amino-5-cyano-6-ethoxy-2-pyridinyl)-2,5-dimethoxy-4-(methylsulfonyl)-
Canonical SMILESCCOc1nc(NC(=O)Cc2cc(OC)c(S(C)(=O)=O)cc2OC)cc(N)c1C#N
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.82
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 8.3 Ki ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 8.1 Ki ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 7.1 Ki ChEMBL;BindingDB