Molecule Details
InChIKeyUILRVXAQZKZLBN-UHFFFAOYSA-N
Compound NameN-[2-methyl-4-(1-methyl-4,10-dihydropyrazolo[4,5-c][1,5]benzodiazepine-5-carbonyl)phenyl]-2-phenylbenzamide
Canonical SMILESCc1cc(C(=O)N2Cc3cnn(C)c3Nc3ccccc32)ccc1NC(=O)c1ccccc1-c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.53
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30518 AVPR2 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P37288 AVPR1A Homo sapiens Human PF00001 PF08983 7.4 Ki ChEMBL;BindingDB
P30559 OXTR Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB