Molecule Details
InChIKeyUIEXDKQSWATHMD-UHFFFAOYSA-N
Compound NameN-(3,4-Dimethoxyphenyl)-2-(1h-Pyrazol-4-Yl)-1h-Pyrrolo[3,2-C]pyridin-6-Amine
Canonical SMILESCOc1ccc(Nc2cc3[nH]c(-c4cn[nH]c4)cc3cn2)cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.45
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P33981 TTK Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
P20248 CCNA2 Homo sapiens Human PF02984 PF00134 PF16500 7.4 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB