Molecule Details
InChIKeyUIAYVIIHMORPSJ-UHFFFAOYSA-N
Canonical SMILESCN(C(=O)CCCOc1ccc2[nH]c(=O)ccc2c1)C1CCCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.73
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB19897
Drug NameCilostamide
CAS Number68550-75-4
Groups experimental
ATC Codes nan
DescriptionCilostamide is a small molecule drug. Cilostamide has a monoisotopic molecular weight of 342.19 Da.

Categories: Antiplatelet agents Enzyme Inhibitors Hematologic Agents Heterocyclic Compounds, Fused-Ring Phosphodiesterase Inhibitors Quinolines
Cross-references: BindingDB: 50027177 ChEBI: 92503 CHEMBL34431 ZINC: ZINC000003872076
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q14432 PDE3A Homo sapiens Human PF00233 7.8 IC50 ChEMBL;BindingDB
Q13370 PDE3B Homo sapiens Human PF00233 7.7 IC50 ChEMBL;BindingDB