Molecule Details
InChIKeyUIAPXMIGDHYZKN-UHFFFAOYSA-N
Canonical SMILESO=C1CCC2(CN(Cc3ccc(-c4cccc(-c5cccc(-c6ccc(CN7CC8(CCC(=O)N8)C7)c(F)n6)c5Cl)c4Cl)nc3F)C2)N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9BQ51 PDCD1LG2 Homo sapiens Human PF22705 6.1 IC50 ChEMBL;BindingDB
Q9NZQ7 CD274 Homo sapiens Human PF08205 PF07686 6.1 IC50 ChEMBL