Molecule Details
InChIKeyUHXVRMFFZLLZNC-UHFFFAOYSA-N
Compound Name3-[3-[4-(1-Aminocyclobutyl)phenyl]-5-(3-aminophenyl)imidazo[4,5-b]pyridin-2-yl]pyridin-2-amine
Canonical SMILESNc1cccc(-c2ccc3nc(-c4cccnc4N)n(-c4ccc(C5(N)CCC5)cc4)c3n2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31749 AKT1 Homo sapiens Human PF00169 PF00069 PF00433 8.7 IC50 ChEMBL;BindingDB
P31751 AKT2 Homo sapiens Human PF00169 PF00069 PF00433 8.4 IC50 ChEMBL;BindingDB
Q9Y243 AKT3 Homo sapiens Human PF00169 PF00069 PF00433 8.2 IC50 ChEMBL;BindingDB