Molecule Details
InChIKeyUHWZHRQDJOKBQY-UHFFFAOYSA-N
Compound Name4-methyl-3-(2-pyrazolo[1,5-a]pyrimidin-6-ylethynyl)-N-[3-(pyrrolidin-1-ylmethyl)-5-(trifluoromethyl)phenyl]benzamide
Canonical SMILESCc1ccc(C(=O)Nc2cc(CN3CCCC3)cc(C(F)(F)F)c2)cc1C#Cc1cnc2ccnn2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.97
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q08345 DDR1 Homo sapiens Human PF21114 PF00754 PF07714 7.9 IC50 ChEMBL;BindingDB
Q16832 DDR2 Homo sapiens Human PF21114 PF00754 PF07714 6.9 IC50 ChEMBL;BindingDB
P10721 KIT Homo sapiens Human PF00047 PF07714 6.1 IC50 ChEMBL;BindingDB