Molecule Details
InChIKeyUHWVXMZHHQZRCC-UHFFFAOYSA-N
Compound Name2-Methyl-2-[[[5-[[6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino]-3-isothiazolyl]methyl](2,2,2-trifluoroethyl)amino]-1-propanol Hydrochloride
Canonical SMILESCc1cn2c(-c3cn[nH]c3)cnc2c(Nc2cc(CN(CC(F)(F)F)C(C)(C)CO)ns2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.55
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O75716 STK16 Homo sapiens Human PF00069 8.4 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB