Molecule Details
InChIKeyUGTWRNKTBHMJMC-UHFFFAOYSA-N
Compound Name1-Ethyl-3-[3-[[1-[2-(2-methylquinolin-5-yl)oxyethyl]piperidin-4-yl]methyl]phenyl]urea
Canonical SMILESCCNC(=O)Nc1cccc(CC2CCN(CCOc3cccc4nc(C)ccc34)CC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 9.6 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 7.6 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB