Molecule Details
InChIKeyUGLMDRPTTBWXIB-UHFFFAOYSA-N
Compound Name8-[5-(trifluoromethyl)-1H-pyrazol-4-yl]-5lambda4-thia-9,14,15-triazatetracyclo[8.7.0.02,7.013,17]heptadeca-1(10),2(7),8,11,13(17),15-hexaene 5-oxide
Canonical SMILES[O-][S+]1CCc2c(c(-c3c[nH]nc3C(F)(F)F)nc3ccc4[nH]ncc4c23)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.52
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 7.8 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
P78396 CCNA1 Homo sapiens Human PF02984 PF00134 PF16500 7.4 IC50 ChEMBL