Molecule Details
InChIKeyUGKKDOKVLSCRFL-UHFFFAOYSA-N
Compound Name4-Amino-5-chloro-6-isopropoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamide
Canonical SMILESCC(C)Oc1nc(C(=O)NCc2ccc(S(C)(=O)=O)cc2)cc(N)c1Cl
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.89
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45984 MAPK9 Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.4 IC50 ChEMBL