Molecule Details
InChIKeyUGDNJOZZYFGNIL-UHFFFAOYSA-N
Compound Name6-amino-N-[4-[[3-[[5-(trifluoromethyl)-2-pyridyl]oxy]-phenyl]methylene]cyclohexyl]pyridine-3-carboxamide
Canonical SMILESNc1ccc(C(=O)NC2CCC(=Cc3cccc(Oc4ccc(C(F)(F)F)cn4)c3)CC2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11712 CYP2C9 Homo sapiens Human PF00067 8.5 IC50 ChEMBL
O00519 FAAH Homo sapiens Human PF01425 8.3 IC50 ChEMBL;BindingDB
P33261 CYP2C19 Homo sapiens Human PF00067 8.0 IC50 ChEMBL