Molecule Details
InChIKeyUFPKGRZJBZMOLS-UHFFFAOYSA-N
Compound Name1-[(3,4-difluorophenyl)methyl]-N-[[6-(3,3-difluoropyrrolidin-1-yl)-3-pyridinyl]methyl]pyrazole-3-carboxamide
Canonical SMILESO=C(NCc1ccc(N2CCC(F)(F)C2)nc1)c1ccn(Cc2ccc(F)c(F)c2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43497 CACNA1G Homo sapiens Human PF00520 8.2 IC50 ChEMBL;BindingDB
Q9P0X4 CACNA1I Homo sapiens Human PF00520 8.0 IC50 ChEMBL;BindingDB
O95180 CACNA1H Homo sapiens Human PF00520 7.5 IC50 ChEMBL;BindingDB