Molecule Details
InChIKeyUEYQVGAFBVFHAU-UHFFFAOYSA-N
Compound Name2-N-(3H-benzimidazol-5-yl)-4-N-(2-chlorophenyl)-5-(trifluoromethyl)pyrimidine-2,4-diamine
Canonical SMILESFC(F)(F)c1cnc(Nc2ccc3[nH]cnc3c2)nc1Nc1ccccc1Cl
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.87
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P06493 CDK1 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
P11802 CDK4 Homo sapiens Human PF00069 8.9 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 8.7 pIC50 TTD_MultiTarget