Molecule Details
InChIKeyUEUUWJVQGWZIJY-UHFFFAOYSA-N
Compound Name4-chloro-N-(6-pyrimidin-5-yloxypyrazin-2-yl)pyridine-2-carboxamide
Canonical SMILESO=C(Nc1cncc(Oc2cncnc2)n1)c1cc(Cl)ccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.64
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P41594 GRM5 Homo sapiens Human PF00003 PF01094 PF10606 PF07562 7.1 IC50 ChEMBL;BindingDB
P05177 CYP1A2 Homo sapiens Human PF00067 6.2 IC50 ChEMBL;BindingDB