Molecule Details
InChIKeyUDUOGLZZYDDSKR-UHFFFAOYSA-N
Compound Name5-phenyl-N-(4-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)butyl)pyridin-2-amine
Canonical SMILESFC(F)(F)c1cccc(N2CCN(CCCCNc3ccc(-c4ccccc4)cn3)CC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.48
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P35348 ADRA1A Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB