Molecule Details
InChIKeyUDOITUAULPBVSE-UHFFFAOYSA-N
Compound NameN-(4-(methylsulfonyl)benzyl)-4-amino-5-cyano-6-isopropoxypicolinamide
Canonical SMILESCC(C)Oc1nc(C(=O)NCc2ccc([S@SP2](C)(=O)=O)cc2)cc(N)c1C#N
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.28
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.6 IC50 ChEMBL