Molecule Details
InChIKeyUDCDKGHUDICLCJ-LRDDRELGSA-N
Compound Name(S)-3-Phenyl-2-[(S)-2-(4-sulfamoyl-benzoylamino)-propionylamino]-propionic acid
Canonical SMILESC[C@H](NC(=O)c1ccc(S(N)(=O)=O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.45
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 7.9 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.9 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 6.5 Ki ChEMBL;BindingDB