Molecule Details
InChIKeyUCPDUMRVOIJGJU-UHFFFAOYSA-N
Compound NameN-ethyl-2-(2-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinazolin-4-yl]amino}-1,3-thiazol-5-yl)-N-phenylacetamide
Canonical SMILESCCN(C(=O)Cc1cnc(Nc2ncnc3cc(OCCCN4CCOCC4)c(OC)cc23)s1)c1ccccc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.26
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 7.3 pIC50 TTD_MultiTarget