Molecule Details
InChIKeyUBQAXNUSTYBVJI-UHFFFAOYSA-N
Compound Namen-(4-Methyl-3-(3-methyl-1h-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(quinoxalin-5-yl)acetamide
Canonical SMILESCc1n[nH]c(-c2c(C)csc2NC(=O)Cc2cccc3nccnc23)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.47
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45984 MAPK9 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB