Molecule Details
InChIKeyUBNQUXARYFJNPF-UHFFFAOYSA-N
Compound Name4-[6-fluoro-2-[5-[(sulfamoylamino)methyl]-1,3,4-oxadiazole-2-carbonyl]-1,3-benzothiazol-5-yl]-N-(2,2,2-trifluoroethyl)benzamide
Canonical SMILESNS(=O)(=O)NCc1nnc(C(=O)c2nc3cc(-c4ccc(C(=O)NCC(F)(F)F)cc4)c(F)cc3s2)o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11150 LIPC Homo sapiens Human PF00151 PF01477 8.4 IC50 ChEMBL;BindingDB
Q9Y5X9 LIPG Homo sapiens Human PF00151 PF01477 6.7 IC50 ChEMBL;BindingDB