Molecule Details
InChIKeyUBBCZBKJYNXHGT-GFCCVEGCSA-N
Compound NameN~2~-(1-Cyclopentyl-4-Oxo-4,7-Dihydro-1h-Pyrazolo[3,4-D]pyrimidin-6-Yl)-N-(4-Methoxyphenyl)-D-Alaninamide
Canonical SMILESCOc1ccc(NC(=O)[C@@H](C)Nc2nc3c(cnn3C3CCCC3)c(=O)[nH]2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.53
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O76083 PDE9A Homo sapiens Human PF00233 9.2 IC50 ChEMBL;BindingDB
O76074 PDE5A Homo sapiens Human PF01590 PF00233 7.0 IC50 ChEMBL;BindingDB
Q01064 PDE1B Homo sapiens Human PF00233 PF08499 6.3 IC50 ChEMBL;BindingDB