Molecule Details
InChIKeyUAILHDKDBBFHDN-STWLFGJUSA-M
Compound Name(5R),(6E)-6-(5,6-dihydro-8H-imidazo[2,1-c][1,4]thiazin-2-ylmethylene)-7-oxo-4-thia-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid sodium salt
Canonical SMILESO=C([O-])C1=CS[C@@H]2/C(=C/c3cn4c(n3)CSCC4)C(=O)N12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Unknown
Avg pChEMBL6.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P25910 ccrA Bacteroides fragilis Pathogen 7.0 IC50 ChEMBL;BindingDB
P05364 ampC Enterobacter cloacae Pathogen PF00144 6.4 IC50 ChEMBL;BindingDB
P62593 bla Escherichia coli Pathogen PF13354 6.1 IC50 ChEMBL;BindingDB