Molecule Details
InChIKeyTZISXJSUKNYDMP-LLVKDONJSA-N
Compound Name6-(2-aminoethylsulfonyl)-3-[2-[(1S)-1-amino-2-hydroxyethyl]-1H-benzimidazol-4-yl]-2-(2H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESNCCS(=O)(=O)c1ccc(-c2cccc3[nH]c([C@H](N)CO)nc23)c(-c2nn[nH]n2)c1S(N)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.22
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 9.6 IC50 BindingDB
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.4 IC50 ChEMBL;BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.7 IC50 BindingDB