Molecule Details
InChIKeyTZIIUZZREBUIBM-UHFFFAOYSA-N
Compound Name3-(4-(3-Fluoro-2-(trifluoromethyl)phenyl)piperidine-1-carbonyl)-[1,2,4]triazolo[4,3-a]pyridine-6-carbonitrile
Canonical SMILESN#Cc1ccc2nnc(C(=O)N3CCC(c4cccc(F)c4C(F)(F)F)CC3)n2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.44
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P02753 RBP4 Homo sapiens Human PF00061 8.3 IC50 ChEMBL;BindingDB
P02766 TTR Homo sapiens Human PF00576 7.9 IC50 BindingDB
P10635 CYP2D6 Homo sapiens Human PF00067 6.1 Ki ChEMBL;BindingDB