Molecule Details
InChIKeyTZFIMSYOLCBXAQ-MDZDMXLPSA-N
Compound Name3-[[(E)-3-(1-methyl-[1,3]thiazolo[3,2-a]benzimidazol-2-yl)-3-oxoprop-1-enyl]amino]benzenesulfonamide
Canonical SMILESCc1c(C(=O)/C=C/Nc2cccc(S(N)(=O)=O)c2)sc2nc3ccccc3n12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.37
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43570 CA12 Homo sapiens Human PF00194 6.6 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 6.4 Ki ChEMBL;BindingDB
Q16790 CA9 Homo sapiens Human PF00194 6.1 Ki ChEMBL;BindingDB