Molecule Details
InChIKeyTZDWHPRZIBFLNB-UHFFFAOYSA-N
Compound NameN-[4-cyano-1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-(1-methylindazol-5-yl)acetamide
Canonical SMILESCn1ncc2cc(CC(=O)Nc3nn(Cc4ccc(F)c(F)c4)cc3C#N)ccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.82
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9P0X4 CACNA1I Homo sapiens Human PF00520 8.0 IC50 ChEMBL;BindingDB
O43497 CACNA1G Homo sapiens Human PF00520 7.8 IC50 ChEMBL;BindingDB
O95180 CACNA1H Homo sapiens Human PF00520 7.7 IC50 ChEMBL;BindingDB