Molecule Details
InChIKeyTYOXFTVBALRDRN-UHFFFAOYSA-N
Compound NameUS11066396, Example 261
Canonical SMILESFc1ccc2ccc(OCc3ccc(-c4noc(C(F)(F)F)n4)c(F)c3)nc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.08
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UQL6 HDAC5 Homo sapiens Human PF12203 PF00850 7.6 IC50 ChEMBL;BindingDB
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 7.5 IC50 ChEMBL;BindingDB
Q13547 HDAC1 Homo sapiens Human PF00850 6.1 IC50 ChEMBL;BindingDB