Molecule Details
InChIKeyTYGGQOXANGOHKM-UHFFFAOYSA-N
Compound Name2-(5-{3,5-Bis[5-(isoquinolin-2-ium-2-yl)pentyl]phenyl}pentyl)isoquinolin-2-ium tribromide
Canonical SMILESc1ccc2c[n+](CCCCCc3cc(CCCCC[n+]4ccc5ccccc5c4)cc(CCCCC[n+]4ccc5ccccc5c4)c3)ccc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.97
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9GZZ6 CHRNA10 Homo sapiens Human PF02931 PF02932 8.4 IC50 ChEMBL;BindingDB
Q9UGM1 CHRNA9 Homo sapiens Human PF02931 PF02932 8.4 IC50 ChEMBL
P36544 CHRNA7 Homo sapiens Human PF02931 PF02932 7.0 IC50 ChEMBL;BindingDB