Molecule Details
InChIKeyTYFFXNLNRYRUAU-LFSOJSGESA-N
Compound Namec[Nle-Nle-D-Nal(2')-Arg-Trp-Glu]-NH2
Canonical SMILESCCCC[C@@H]1NC(=O)CC[C@@H](C(N)=O)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H](Cc2ccc3ccccc3c2)NC(=O)[C@H](CCCC)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P33032 MC5R Homo sapiens Human PF00001 8.4 IC50 ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 8.2 IC50 ChEMBL;BindingDB
P32245 MC4R Homo sapiens Human PF00001 7.8 IC50 ChEMBL;BindingDB