Molecule Details
InChIKeyTYBHAECIGHGJDF-UHFFFAOYSA-N
Canonical SMILESCOc1cc(Nc2nccc(Oc3ccc(NC(=O)Nc4cc(C(C)C)nn4-c4ccc(C)c(C)c4)c4ccccc34)n2)cc(C(=O)NCCN2CCOCC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.11
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 8.3 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 7.9 IC50 ChEMBL;BindingDB