Molecule Details
InChIKeyTXMPFIFVHHJTKU-UHFFFAOYSA-N
Compound Name3-(3-amino-2H-indazol-6-yl)-2-(1H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESNc1[nH]nc2cc(-c3cccc(S(N)(=O)=O)c3-c3nnn[nH]3)ccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.88
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.2 IC50 ChEMBL;BindingDB
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 7.8 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 6.7 IC50 BindingDB